|
|
|
篇目详细内容 |
|
【篇名】 |
Synthesis and fungicidal activity of novel 3,5-diarylpyrazole derivatives |
|
【刊名】 |
Frontiers of Chemistry in China |
|
【刊名缩写】 |
Front. Chem. China |
|
【ISSN】 |
1673-3495 |
|
【EISSN】 |
1673-3614 |
|
【DOI】 |
10.1007/s11458-008-0075-3 |
|
【出版社】 |
Higher Education Press and Springer-Verlag |
|
【出版年】 |
2008 |
|
【卷期】 |
3
卷4期 |
|
【页码】 |
418-421
页,共
4
页 |
|
【作者】 |
LIU Xinhua;
ZHU Jing;
PAN Chunxiu;
LI Bo;
SONG Bao‘an;
|
|
【关键词】 |
2-chlorobenzaldehyde; 3,5-diarylpyrazole; synthesis; fungicide |
【摘要】 |
|
(E)-3-(2-chlorophenyl)-1-(2,4-dichlorophenyl)prop-2-en-1-one was prepared from 2-chlorobenzaldehyde followed by cyclization with hydrazine monohydrate. Eight new 3-(2,4-Di-chlorophenyl)-5-(2-chlorophenyl)-4,5- dihydro-N-acylpyrazole derivatives were synthesized and characterized by elemental analysis, IR and 1H NMR spectroscopy. The experimental results show that the inhibition ratio of compounds 3f towards H. Oryzae and P. oryzae at 50 mg·L-1 is 55.2% and 57.1%, respectively. The inhibition ratio of compounds 3g towards H. Oryzae, P. oryza, S. Sclerotiorum at 50 mg·L-1 is 53.3%, 60.0%, 50.4% respectively. |
|
